SCHEMBL16082245

SCHEMBL16082245

O=C(CO)Nc1ccc2c(c1)CC(Nc1ncnc3ccccc13)C2

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.45
GRM1 Q13255 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
EGFR P00533 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
PDGFRB P09619 1/20 0.42
KIT P10721 1/20 0.42
FLT1 P17948 1/20 0.42
FLT4 P35916 1/20 0.42
KDR P35968 1/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
PARP1 P09874 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16082203 0.87 ABCG2 (0.58) ABCG2EGFRADORA3PDGFRBKIT
SCHEMBL16082987 0.87 ROCK2 (0.42) GRM1EGFRALDH1A1
SCHEMBL16082989 0.87 KDR (0.41) GRM1EGFRPDGFRBKITFLT1
SCHEMBL16082747 0.87 EGFR (0.46) GRM1EGFR
SCHEMBL16082719 0.80 EGFR (0.45) EGFR
SCHEMBL16082966 0.78 EGFR (0.52) EGFR
SCHEMBL16082332 0.78 EGFR (0.45) EGFR
SCHEMBL9040263 0.78 GBA1 (0.58) GBA1
SCHEMBL16082243 0.78 EGFR (0.54) EGFRPDGFRBPOLB
SCHEMBL16082528 0.77 IRAK4 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014145512-A2 POTENT SMALL MOLECULE INHIBITORS OF AUTOPHAGY, AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2014-09-18 WO disclosed