Mg-132

Mg-132

SCHEMBL160925

CC(C)C[C@@H](C=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.77
PSMB5 P28074 1/20 0.77
PSMB2 P49721 1/20 0.77
CTSL P07711 9/20 0.72
CTSB P07858 6/20 0.72
CTSK P43235 5/20 0.69
CTSS P25774 2/20 0.65
CAPN1 P07384 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mg-132 SCHEMBL13436259 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL7862424 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL10006388 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL14579851 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL2522088 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL5062219 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL2535252 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
Mg-132 SCHEMBL14514061 1.00 PSMB1 (0.77) PSMB1PSMB5PSMB2CTSLCTSB
SCHEMBL7710728 0.99 PSMB1 (0.78) PSMB1PSMB5PSMB2CTSLCTSB
SCHEMBL3054703 0.99 PSMB1 (0.78) PSMB1PSMB5PSMB2CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4392 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
US-20260102417-A1 COMPOSITIONS FOR THE TREATMENT AND PREVENTION OF CANCER KEYZELL HOLDING S L (ES) 2026-04-16 US claimed
US-20260069567-A1 Pharmaceutical Combinations For The Treatment Of Cancer PRESAGE BIOSCIENCES, INC. (US) 2026-03-12 US claimed
EP-4706663-A2 FAP-ACTIVATED PROTEASOME INHIBITORS FOR TREATING SOLID TUMORS Trustees Of Tufts College (US) 2026-03-11 EP claimed
US-12529162-B2 Method of screening for peptides capable of binding to a ubiquitin protein ligase (E3) PHOREMOST LIMITED (GB) 2026-01-20 US claimed
EP-4667458-A1 PHARMACEUTICAL COMPOSITION FOR TREATMENT OF CANCER, COMPRISING SOS1 INHIBITOR AND ANTICANCER DRUG Kanaph Therapeutics Inc. (KR) 2025-12-24 EP claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US claimed
US-20250367304-A1 FAP-ACTIVATED PROTEASOME INHIBITORS FOR TREATING SOLID TUMORS TUFTS COLLEGE (US) 2025-12-04 US claimed
EP-4648769-A2 NECROSIS INHIBITOR Linkgevity Limited (GB) 2025-11-19 EP claimed
EP-3436002-B1 PHARMACEUTICAL COMBINATIONS FOR THE TREATMENT OF CANCER PRESAGE BIOSCIENCES INC (US) 2025-11-05 EP claimed
WO-2004004749-A1 PROTEASEOME INHIBITORS FOR THE TREATMENT OF HERPESVIRIDAE INFECTED INDIVIDUALS CHARITE - UNIVERSITÄTSMEDIZIN BERLIN (DE) 2004-01-15 WO claimed
WO-2002101012-A9 REGULATION OF TRANSGENE EXPRESSION FOLLOWING AAV TRANSDUCTION CHILDREN S HOSPITAL RES FOUNDA (US) 2003-12-18 WO claimed
WO-2003084551-A1 AGENTS FOR TREATING FLAVIVIRIDAE INFECTIONS VIROMICS GMBH (DE) 2003-10-16 WO claimed
WO-2003064453-A2 TROJAN INHIBITORS, METHOD FOR THE PRODUCTION AND USE THEREOF VIROMICS GMBH (DE) 2003-08-07 WO claimed
EP-1326632-A2 AGENTS FOR THE TREATMENT OF VIRAL INFECTIONS VIROMICS GMBH (DE) 2003-07-16 EP claimed
US-20030003583-A1 Regulation of transgene expression following AAV transduction CHILDREN'S HOSPITAL RESEARCH FOUNDATION 2003-01-02 US claimed
WO-2002101012-A2 REGULATION OF TRANSGENE EXPRESSION FOLLOWING AAV TRANSDUCTION CHILDREN'S HOSPITAL RESEARCH FOUNDATION (US) 2002-12-19 WO claimed
US-20020111314-A1 Novel stimulation of gene expression and protein synthesis of heat shock protein 72/73 (Hsp 70) THE TRUSTEES OF COLUMBIA UNIVERSITY (US) 2002-08-15 US claimed
WO-2002030455-A2 AGENTS FOR THE TREATMENT OF VIRAL INFECTIONS VIROMICS GMBH (DE) 2002-04-18 WO claimed
US-5942494-A Stimulation of gene expression and synthesis of heat shock protein 72/73 (HSP 70) THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1999-08-24 US claimed