SCHEMBL16098685

SCHEMBL16098685

Oc1ccc2c3cc(CF)ncc3n(CCN3CCOCC3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 6/20 0.40
WEE1 P30291 6/20 0.40
CNR2 P34972 3/20 0.40
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
TSHR P16473 3/20 0.37
POLB P06746 1/20 0.37
SRC P12931 1/20 0.36
MAPT P10636 3/20 0.36
MAPK1 P28482 2/20 0.36
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
ALOX15 P16050 1/20 0.35
LMNA P02545 1/20 0.35
CREBBP Q92793 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16099437 0.90 NPY5R (0.38) CNR2ESR1ESR2POLB
SCHEMBL16098994 0.88 XDH (0.37) CHEK1WEE1CNR2CDK1CCNB1
SCHEMBL16093856 0.80 ATM (0.36) CNR2TSHRMAPTATMALOX15
SCHEMBL16099208 0.78 WEE1 (0.41) CHEK1WEE1ESR1ESR2POLB
SCHEMBL30940010 0.72 DYRK1A (0.48)
SCHEMBL16099657 0.72 DYRK1A (0.48)
SCHEMBL16123614 0.72 HASPIN (0.47) CHEK1WEE1CNR2ESR1ESR2
SCHEMBL30939941 0.72 HASPIN (0.47) CHEK1WEE1CNR2ESR1ESR2
SCHEMBL23234240 0.70 ALDH1A1 (0.46) CNR2TSHRTP53LMNAKDM4E
SCHEMBL16123513 0.70 CNR2 (0.41) CNR2TSHRMAPTTP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968284-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH Osteoqc Inc. (CA) 2016-01-20 EP disclosed
WO-2014153203-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH OSSIFI INC. (US) 2014-09-25 WO disclosed