SCHEMBL160987

SCHEMBL160987

O=C(Nc1ccc(-c2cnc(C3CCNCC3)s2)cc1)Nc1ccc(F)cc1F

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.59
HTT P42858 2/20 0.47
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
PIK3CA P42336 1/20 0.44
MTOR P42345 1/20 0.44
PIK3CG P48736 1/20 0.44
MAPT P10636 2/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
LMNA P02545 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL162765 0.99 DGAT1 (0.59) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL163112 0.90 DGAT1 (0.58) DGAT1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL164216 0.90 DGAT1 (0.57) DGAT1CA12CA1CA2CA9
SCHEMBL164677 0.88 DGAT1 (0.73) DGAT1HTTNPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL160909 0.88 DGAT1 (0.57) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL158343 0.85 DGAT1 (0.56) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL161308 0.85 DGAT1 (0.61) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL164678 0.85 DGAT1 (0.56) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL162343 0.85 DGAT1 (0.56) DGAT1HTTNPC1RAB9ASMN1; SMN2
SCHEMBL161999 0.85 DGAT1 (0.58) DGAT1HTTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed