SCHEMBL163112

SCHEMBL163112

O=C(Nc1ccc(-c2cnc(C3CCNCC3)s2)cc1)Nc1cc(F)c(F)cc1F

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 7/20 0.58
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
CTSC P53634 1/20 0.40
MAP4K3 Q8IVH8 2/20 0.39
DYRK1A Q13627 2/20 0.38
WNT1 P04628 1/20 0.38
GSK3B P49841 1/20 0.38
JAK3 P52333 1/20 0.38
SNCA P37840 1/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL164216 0.99 DGAT1 (0.57) DGAT1CA12CA1CA2CA9
SCHEMBL160987 0.90 DGAT1 (0.59) DGAT1CA12CA1CA2CA9
SCHEMBL173959 0.90 DGAT1 (0.60) DGAT1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL162765 0.90 DGAT1 (0.59) DGAT1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL160909 0.87 DGAT1 (0.57) DGAT1CA12CA1CA2CA9
SCHEMBL165743 0.87 DGAT1 (0.73) DGAT1CA12CA1CA2CA9
SCHEMBL162997 0.85 DGAT1 (0.55) DGAT1CA12CA1CA2CA9
SCHEMBL160661 0.85 DGAT1 (0.59) DGAT1CA12CA1CA2CA9
SCHEMBL162202 0.85 DGAT1 (0.57) DGAT1CA12CA1CA2CA9
SCHEMBL15022085 0.85 DGAT1 (0.55) DGAT1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed