SCHEMBL16099720

SCHEMBL16099720

C1CC2CCCC(C1)C2.c1ccc2c(c1)C1CCC2C1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
PDPK1 O15530 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
IDO1 P14902 2/20 0.33
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC18A3 Q16572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913571 0.85 CHRNB4 (0.54) CHRNB4CHRNA3PDPK1NOS3NOS1
SCHEMBL30166929 0.85 CHRNB4 (0.59) CHRNB4CHRNA3PDPK1IDO1CHRNB2
SCHEMBL221689 0.85 CHRNB4 (0.59) CHRNB4CHRNA3PDPK1IDO1CHRNB2
SCHEMBL23797352 0.85 CHRNB4 (0.59) CHRNB4CHRNA3PDPK1IDO1CHRNB2
SCHEMBL11704162 0.80 CHRNB4 (0.54) CHRNB4CHRNA3PDPK1NOS1
SCHEMBL11701290 0.78 CHRNB4 (0.52) CHRNB4CHRNA3NOS1SLC18A3
SCHEMBL11704954 0.78 CHRNB4 (0.52) CHRNB4CHRNA3NOS1SLC18A3
SCHEMBL2913620 0.78 CHRNB4 (0.44) CHRNB4CHRNA3PDPK1IDO1NOS3
SCHEMBL6940509 0.74 CHRNB4 (0.50) CHRNB4CHRNA3PDPK1IDO1CHRNB2
SCHEMBL3425103 0.74 CHRNB4 (0.50) CHRNB4CHRNA3PDPK1IDO1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968280-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND METHODS OF USE THEREOF Genentech, Inc. (US) 2016-01-20 EP disclosed
WO-2014153037-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-09-25 WO disclosed