SCHEMBL16104161

SCHEMBL16104161

NC(=O)[C@@H]1CC[C@@H]2CCCC[C@H](N)C(=O)N21

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XIAP P98170 6/20 0.36
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.35
APEX1 P27695 1/20 0.35
F2 P00734 1/20 0.34
PLG P00747 1/20 0.34
BIRC3 Q13489 1/20 0.33
BIRC2 Q13490 1/20 0.33
BIRC8 Q96P09 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9609009 0.97 F2 (0.36) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL14140109 0.92 CYP3A4 (0.36) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL5832039 0.87 XIAP (0.38) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL5832021 0.87 XIAP (0.38) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL8358700 0.87 XIAP (0.38) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL9609014 0.83 ACE (0.40) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL10331862 0.83 ACE (0.40) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL26256186 0.83 ACE (0.40) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL12034318 0.83 ACE (0.40) XIAPCYP3A4TSHRTDP1MAPT
SCHEMBL13259956 0.82 F2 (0.38) XIAPCYP3A4TSHRTDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019671-B1 INTERMEDIATES FOR THE PREPARATION OF BIVALENT SMAC MIMETICS UNIV MICHIGAN (US) 2014-09-24 EP disclosed