SCHEMBL1610598

SCHEMBL1610598

CCC/C=[C]\c1cccc2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHAT P28329 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP2A6 P11509 2/20 0.36
GRM5 P41594 1/20 0.36
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR1B P28222 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
HSD17B10 Q99714 2/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HPGD P15428 1/20 0.33
EPHX1 P07099 1/20 0.33
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27293170 0.90 HTR1B (0.37) CHATCA1CA2ALDH1A1CYP2A6
SCHEMBL1609445 0.90 HTR1B (0.37) CHATCA1CA2ALDH1A1CYP2A6
SCHEMBL1610676 0.88 CNR1 (0.38) CHATALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL1612559 0.87 CHAT (0.40) CHATALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL1609453 0.86 ALDH1A1 (0.34) ALDH1A1CYP2A6CYP1A2SIGMAR1HSD17B10
SCHEMBL1611479 0.85 CHAT (0.40) CHATCA1CA2ALDH1A1CYP2A6
SCHEMBL1611797 0.77 MEN1 (0.35) ALDH1A1CYP1A2CYP2D6TDP1
SCHEMBL1609255 0.76 NR1I2 (0.39) ALDH1A1CYP2A6CYP1A2CYP2C19HSD17B10
SCHEMBL1610267 0.76 MAPT (0.35) CHATALDH1A1CYP2D6
SCHEMBL1612130 0.76 TSHR (0.43) ALDH1A1GRM5TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110087034-A1 Organic Semiconductor Material SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2011-04-14 US disclosed
EP-2248818-A1 ORGANIC SEMICONDUCTOR MATERIAL Sumitomo Chemical Company, Limited (JP) 2010-11-10 EP disclosed
US-7557127-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2009-07-07 US disclosed
US-20090054464-A1 HDAC INHIBITOR ASTELLAS PHARMA INC. (JP) 2009-02-26 US disclosed
US-7465731-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2008-12-16 US disclosed
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
US-20060052599-A1 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2006-03-09 US disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed
EP-0602242-A1 BENZISOXAZOLE COMPOUND AND USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-06-22 EP disclosed
EP-0498680-A1 New beta-amino-alpha-hydroxycarboxylic acids and their use Sankyo Company Limited (JP) 1992-08-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052599-A1 HDAC inhibitor HDAC1, HDAC2, HDAC11 CHAT 2847/4885CA1 2168/4885CA2 1328/4885
US-20090054464-A1 HDAC INHIBITOR HDAC1, HDAC2, HDAC8 CHAT 3056/4885CA1 2348/4885CA2 1794/4885
US-20110087034-A1 Organic Semiconductor Material OR10J3, TST, OR51E2 CHAT 1928/4885CA1 3989/4885CA2 3911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.