SCHEMBL16147805

SCHEMBL16147805

N#Cc1cc2ccccc2c(OCC2CCCN2C(=O)O)n1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.51
IRAK4 Q9NWZ3 3/20 0.43
PREP P48147 4/20 0.41
DPP4 P27487 5/20 0.41
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38
KDM2B Q8NHM5 2/20 0.37
DPP8 Q6V1X1 2/20 0.37
DPP9 Q86TI2 2/20 0.37
DPP7 Q9UHL4 2/20 0.37
FAP Q12884 1/20 0.37
CYP2D6 P10635 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
FAAH O00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16008123 0.86 BTK (0.47) BTKIRAK4DPP4
SCHEMBL16008653 0.86 BTK (0.47) BTKIRAK4DPP4
SCHEMBL16008121 0.86 BTK (0.47) BTKIRAK4DPP4
SCHEMBL18455650 0.83 BTK (0.44) BTKIRAK4PREPDPP4HCRTR1
SCHEMBL4140738 0.73 ABHD6 (0.54) DPP4
SCHEMBL15811746 0.73 ABHD6 (0.54) DPP4
SCHEMBL16008553 0.72 BTK (0.50) BTKKDM2B
SCHEMBL5413716 0.72 FFAR1 (0.55)
SCHEMBL3800651 0.71 CPT1A (0.54) DPP4HCRTR1HCRTR2
SCHEMBL29007902 0.70 SSTR4 (0.44) DPP4HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970202-A1 PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2016-01-20 EP disclosed
WO-2014164558-A1 PYRIDINYL AND FUSED PYRIDINYL TRIAZOLONE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-10-09 WO disclosed