SCHEMBL16149558

SCHEMBL16149558

CC(C)(C)N1CCN(C(=O)c2ccc(-c3cnc4ccccc4c3)cc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 2/20 0.69
MKNK2 Q9HBH9 3/20 0.55
MKNK1 Q9BUB5 2/20 0.55
PIK3CA P42336 4/20 0.53
MTOR P42345 3/20 0.52
KCNH2 Q12809 3/20 0.52
PIK3CD O00329 2/20 0.52
PIK3CB P42338 1/20 0.52
PIK3CG P48736 1/20 0.52
USP7 Q93009 1/20 0.50
MAP4K4 O95819 1/20 0.48
CSNK1G2 P78368 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
MAP4K5 Q9Y4K4 1/20 0.48
HPGD P15428 1/20 0.47
POLB P06746 1/20 0.47
ABL1 P00519 2/20 0.46
BCR P11274 2/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16149302 0.87 FASN (0.64) FASNMKNK2MKNK1PIK3CAMTOR
SCHEMBL7722304 0.87 DPP4 (0.54) FASNPIK3CAMTORKCNH2PIK3CD
SCHEMBL17389567 0.82 FASN (1.00) FASNMKNK2MKNK1USP7
SCHEMBL28389740 0.81 FASN (0.71) FASNHPGDPOLBALDH1A1TSHR
SCHEMBL16151082 0.80 FASN (0.64) FASNMKNK2MKNK1PIK3CAMTOR
SCHEMBL17389638 0.80 FASN (0.64) FASNMKNK2MKNK1PIK3CAMTOR
SCHEMBL17389822 0.80 FASN (0.92) FASNMKNK2MKNK1PIK3CAUSP7
SCHEMBL21497426 0.79 FASN (0.76) FASNMKNK2MKNK1PIK3CAMTOR
Trifluoroacetic Acid SCHEMBL16149057 0.79 MKNK1 (0.66) FASNMKNK2MKNK1PIK3CAMTOR
Trifluoroacetic Acid SCHEMBL16150958 0.79 MKNK1 (0.66) FASNMKNK2MKNK1PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014164767-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITION OF FASN FORMA THERAPEUTICS, INC. (US) 2014-10-09 WO disclosed