SCHEMBL16151069

SCHEMBL16151069

Brc1nc2ccc(OCc3ccccc3)cc2s1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.72
CA12 O43570 1/20 0.64
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64
CA7 P43166 1/20 0.64
CA9 Q16790 1/20 0.64
ALOX5 P09917 1/20 0.53
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
SCD O00767 1/20 0.51
MAOB P27338 2/20 0.50
CYP2D6 P10635 1/20 0.49
KCNH2 Q12809 1/20 0.47
MAOA P21397 1/20 0.47
MAPT P10636 3/20 0.46
CSF1R P07333 2/20 0.46
HPGD P15428 2/20 0.46
IP6K1 Q92551 1/20 0.46
ALDH1A1 P00352 1/20 0.45
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3242108 0.85 CYP3A4 (0.67) CYP3A4CA12CA1CA2CA7
SCHEMBL778719 0.84 CYP3A4 (0.71) CYP3A4CA12CA1CA2CA7
SCHEMBL11414056 0.84 CYP3A4 (1.00) CYP3A4CA12CA1CA2CA7
SCHEMBL3235197 0.84 CYP3A4 (0.71) CYP3A4CA12CA1CA2CA7
SCHEMBL27594904 0.82 CYP3A4 (0.64) CYP3A4CA12CA1CA2CA7
SCHEMBL492622 0.81 CYP3A4 (0.66) CYP3A4CA12CA1CA2CA7
SCHEMBL16150510 0.81 CA2 (0.66) CYP3A4CA12CA1CA2CA7
SCHEMBL24133664 0.79 CYP3A4 (0.70) CYP3A4CA12CA1CA2CA7
SCHEMBL10473859 0.79 CA2 (1.00) CYP3A4CA12CA1CA2CA7
SCHEMBL19783432 0.78 KMT2A (0.69) CYP3A4CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2981527-B1 DERIVATIVES OF LUCIFERIN. UNIV COLLEGE CARDIFF CONSULTANTS LTD (GB) 2018-10-31 EP disclosed
EP-2981527-A1 DERIVATIVES OF LUCIFERIN UCL Business Plc. (GB) 2016-02-10 EP disclosed
WO-2014162157-A1 DERIVATIVES OF LUCIFERIN UCL BUSINESS PLC (GB) 2014-10-09 WO disclosed
WO-2014162157-A1 DERIVATIVES OF LUCIFERIN UCL BUSINESS PLC (GB) 2014-10-09 WO disclosed