SCHEMBL16152829

SCHEMBL16152829

CCOC(=O)/C(=C/CC(C)C)CBr

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.41
ALDH1A1 P00352 6/20 0.41
TRPA1 O75762 1/20 0.41
LMNA P02545 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
S1PR4 O95977 1/20 0.39
S1PR1 P21453 1/20 0.39
MAPK1 P28482 1/20 0.39
GLO1 Q04760 1/20 0.36
PTGS2 P35354 1/20 0.34
CYP2C19 P33261 3/20 0.33
CYP2D6 P10635 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28755858 0.86 GRIK1 (0.36) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL16881890 0.81 GRIK1 (0.43) GRIK1MAPT
SCHEMBL5963393 0.81 ALDH1A1 (0.46) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL5963394 0.81 ALDH1A1 (0.46) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL4661706 0.81 GAA (0.47) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL28582961 0.79 CYP2D6 (0.45) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL2226451 0.79 GRIK1 (0.39) GRIK1ALDH1A1LMNANPSR1MEN1
SCHEMBL5963131 0.78 NPSR1 (0.38) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL28072 0.78 NPSR1 (0.38) GRIK1ALDH1A1TRPA1LMNANPSR1
SCHEMBL5963310 0.78 ALDH1A1 (0.43) GRIK1ALDH1A1TRPA1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9073885-B2 Vitamin D3 lactone derivatives TEIJIN PHARMA LIMITED (JP) 2015-07-07 US disclosed
US-9073885-B2 Vitamin D3 lactone derivatives TEIJIN PHARMA LIMITED (JP) 2015-07-07 US disclosed
EP-1589009-B1 VITAMIN D3 LACTONE DERIVATIVE TEIJIN PHARMA LTD (JP) 2014-10-08 EP disclosed