SCHEMBL16164181

SCHEMBL16164181

CC[C@H](NC(=O)O)[C@@H](CC)Nc1nc(Cl)c(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.40
NPSR1 Q6W5P4 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
S1PR3 Q99500 11/20 0.33
S1PR1 P21453 6/20 0.33
S1PR4 O95977 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 2/20 0.33
PGK1 P00558 1/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.32
S1PR2 O95136 1/20 0.32
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16760788 0.91 KHK (0.39) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16165332 0.91 KHK (0.39) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16164780 0.87 KHK (0.35) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16164779 0.87 KHK (0.35) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL14908967 0.85 TRPA1 (0.42) KHK
SCHEMBL16760781 0.85 KHK (0.37) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16760782 0.85 KHK (0.37) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16165734 0.84 KHK (0.38) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL16165736 0.84 KHK (0.38) KHKNPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL14928731 0.83 KHK (0.46) KHKNPSR1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2799431-B1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORP (JP) 2018-01-24 EP disclosed
US-9051310-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2015-06-09 US disclosed
EP-2799431-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM Corporation (JP) 2014-11-05 EP disclosed
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2014-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140309225-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, BTK, NOX4 KHK 1750/4885NPSR1 921/4885CYP1A2 3310/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.