SCHEMBL16166369

SCHEMBL16166369

CC(C)C(=O)Oc1ccc(CO)cc1C(CC(N)(c1ccccc1)C(C)C)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
ALOX15 P16050 2/20 0.42
ADRB2 P07550 1/20 0.39
ADRA2A P08913 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2C P18825 1/20 0.39
DRD1 P21728 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
ELANE P08246 4/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
KIF11 P52732 3/20 0.32
TTR P02766 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982655 0.73 CHRM2 (0.74) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL10098315 0.73 CHRM2 (0.74) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL1116219 0.70 CHRM2 (0.67) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL10098329 0.70 CHRM2 (0.73) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL1116232 0.70 CHRM2 (0.67) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL6757054 0.69 CHRM2 (0.52) CHRM2CHRM1ALOX15ADRB2ADRA2A
Fesoterodine SCHEMBL121127 0.68 CHRM2 (1.00) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL16166473 0.68 CHRM2 (0.70) CHRM2CHRM1ALOX15ADRB2ADRA2A
SCHEMBL724335 0.68 CHRM2 (0.84) CHRM2CHRM1ALOX15ADRB2ADRA2A
Fesoterodine SCHEMBL812986 0.68 CHRM2 (1.00) CHRM2CHRM1ALOX15ADRB2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014167578-A2 NOVEL POLYMORPH OF ISOBUTYRIC ACID 2-((R)-3-DIISOPROPYL AMINO-1-PHENYLPROPYL)-4-(HYDROXYMETHYL)PHENYL ESTER HYDROCHLORIDE AND PROCESS FOR PREPARATION THEREOF MSN LABORATORIES LIMITED (IN) 2014-10-16 WO disclosed