SCHEMBL16175603

SCHEMBL16175603

O=C(NCCc1ccccc1)ON1CCC2(CC1)CC(c1ccccc1)=NO2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
TAAR1 Q96RJ0 2/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
DRD2 P14416 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011475 0.93 TAAR1 (0.47) TAAR1NPC1RAB9APOLB
SCHEMBL16175720 0.93 KMT2A (0.45) KMT2ANPC1RAB9A
SCHEMBL5012262 0.91 NPC1 (0.43) KMT2ATAAR1NPC1GAARAB9A
SCHEMBL5014451 0.91 TP53 (0.43) KMT2ADRD2
SCHEMBL5011116 0.90 ALDH1A1 (0.46) KMT2ATAAR1NPC1GAARAB9A
SCHEMBL5012838 0.90 KMT2A (0.47) KMT2ACYP1A2POLBCYP2C19
SCHEMBL5124305 0.84 ALDH1A1 (0.46) KMT2ADRD2SIGMAR1
SCHEMBL5012210 0.83 ALDH1A1 (0.45) KMT2A
SCHEMBL16175653 0.83 KMT2A (0.56) KMT2AL3MBTL1
SCHEMBL5064863 0.83 KMT2A (0.52) KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888596-B1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS GRUENENTHAL GMBH (DE) 2014-10-22 EP claimed
EP-1888596-B1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS GRUENENTHAL GMBH (DE) 2014-10-22 EP disclosed