SCHEMBL16198364

SCHEMBL16198364

O=C(/C=C/c1ccccc1Cl)CC(=O)/C=C/c1ccccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.68
HDAC8 Q9BY41 1/20 0.68
HDAC6 Q9UBN7 1/20 0.68
GSR P00390 1/20 0.62
NPC1 O15118 5/20 0.62
RAB9A P51151 5/20 0.62
MAPT P10636 4/20 0.62
MAOB P27338 2/20 0.62
BACE1 P56817 2/20 0.61
HPGD P15428 4/20 0.59
LMNA P02545 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
HSP90AA1 P07900 1/20 0.57
MAOA P21397 1/20 0.57
NFE2L2 Q16236 1/20 0.56
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 2/20 0.55
CYP3A4 P08684 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16198365 1.00 HDAC1 (0.68) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL10375439 0.91 HDAC1 (0.58) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL6955272 0.88 NFE2L2 (0.58) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL1646183 0.87 BACE1 (0.74) HDAC1HDAC8HDAC6MAPTMAOB
SCHEMBL1646186 0.87 BACE1 (0.74) HDAC1HDAC8HDAC6MAPTMAOB
SCHEMBL27321841 0.87 SMN1; SMN2 (0.59) HDAC1HDAC8HDAC6GSRNPC1
Hydrochloric Acid SCHEMBL27314775 0.85 SMN1; SMN2 (0.57) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL11546862 0.84 MAPT (0.56) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL22596712 0.83 HDAC1 (0.67) HDAC1HDAC8HDAC6GSRNPC1
SCHEMBL31553473 0.83 GSR (0.79) HDAC1HDAC8HDAC6GSRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014175841-A1 PALLADIUM COMPLEXES OF CURCUMIN AND ITS ANALOGUES AND METHODS OF PREPARATION OF THE SAME UNIVERZITA KOMENSKEHO V BRATISLAVE (SK) 2014-10-30 WO disclosed