SCHEMBL16199043

SCHEMBL16199043

Cn1nc(-c2ncc(F)c(NC3CCC[C@@H](NC(=O)N4CCC(C)(F)C4)C3)n2)c2cccnc21

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.37
HTR3A P46098 2/20 0.35
MGLL Q99685 3/20 0.34
CCND1 P24385 2/20 0.33
CCNT1 O60563 1/20 0.33
CDK4 P11802 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
CDK6 Q00534 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16199103 1.00 PDE5A (0.37) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199044 0.89 CCNT1 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199101 0.89 CCNT1 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199046 0.86 TLR7 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199027 0.86 TLR7 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199104 0.86 TLR7 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199111 0.86 TLR7 (0.38) PDE5AHTR3AMGLLCCND1CCNT1
SCHEMBL16199021 0.85 PDE5A (0.36) PDE5AHTR3AMGLLAURKAAURKB
SCHEMBL16199110 0.85 PDE5A (0.36) PDE5AHTR3AMGLLAURKAAURKB
SCHEMBL16199045 0.85 PDE5A (0.36) PDE5AHTR3AMGLLAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871774-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-28 US disclosed