SCHEMBL16199575

SCHEMBL16199575

CC(C)(C)OC(=O)N1C[C@H]2CC(OS(C)(=O)=O)C[C@@]2(C)C1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.43
NR1H2 P55055 1/20 0.36
EPHX2 P34913 1/20 0.36
GPR119 Q8TDV5 7/20 0.35
RORC P51449 4/20 0.34
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
USP2 O75604 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16233283 1.00 JAK1 (0.43) JAK1NR1H2EPHX2GPR119RORC
SCHEMBL16192117 0.83 VDR (0.33)
SCHEMBL20466988 0.82 EPHX2 (0.36) JAK1NR1H2EPHX2GPR119RORC
SCHEMBL16233317 0.82 JAK1 (0.48) JAK1NR1H2EPHX2RORCCHRM2
SCHEMBL21774462 0.82 JAK1 (0.48) JAK1NR1H2EPHX2RORCCHRM2
SCHEMBL21774461 0.82 JAK1 (0.48) JAK1NR1H2EPHX2RORCCHRM2
SCHEMBL25504041 0.82 JAK1 (0.48) JAK1NR1H2EPHX2RORCCHRM2
SCHEMBL30402248 0.80 JAK1 (0.47) JAK1NR1H2EPHX2RORCUSP2
SCHEMBL24575156 0.78 JAK1 (0.49) JAK1NR1H2EPHX2RORCCHRM2
SCHEMBL30382336 0.78 JAK1 (0.49) JAK1NR1H2EPHX2RORCCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2796460-A1 PYRROLE SIX-MEMBERED HETEROARYL RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICINAL USES THEREOF Jiangsu Hengrui Medicine Co. Ltd. (CN) 2014-10-29 EP disclosed