SCHEMBL16200078

SCHEMBL16200078

Cc1ccc(-c2[nH]nc(C(F)(F)F)c2Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.39
GAA P10253 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 5/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
PRKDC P78527 1/20 0.38
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
ENPP1 P22413 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875478 0.85 NOTUM (0.41) MAPTGAATP53CYP1A2CYP3A4
SCHEMBL2873737 0.85 MAPK1 (0.40) MAPTGAATP53CYP1A2CYP3A4
SCHEMBL2870930 0.83 GAA (0.41) MAPTGAATP53CYP1A2CYP3A4
SCHEMBL2873684 0.83 ENPP1 (0.44) MAPTCYP1A2CYP2C9MAPK1CYP2C19
SCHEMBL8593143 0.77 NPSR1 (0.43) MAPTLMNAMEN1KMT2ANPSR1
SCHEMBL28724767 0.76 GAA (0.44) MAPTGAACYP1A2CYP2C9MAPK1
SCHEMBL2876798 0.73 NT5E (0.42) MAPTTP53MAPK1LMNASMN1; SMN2
SCHEMBL16200084 0.73 CYP2A6 (0.41) CYP1A2CYP3A4SMN1; SMN2ALDH1A1HSD17B10
SCHEMBL8196073 0.71 ENPP1 (0.35) MAPK1LMNAPIK3CDPIK3CAPIK3CB
SCHEMBL6548270 0.71 PTGS2 (0.51) CYP3A4CYP2D6CYP2C9LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed