SCHEMBL16200084

SCHEMBL16200084

FC(F)(F)c1n[nH]c(-c2cccnc2)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
BTK Q06187 1/20 0.40
CYP19A1 P11511 1/20 0.40
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
RAB9A P51151 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2B6 P20813 1/20 0.39
PIM1 P11309 1/20 0.39
NPY5R Q15761 1/20 0.39
IDO1 P14902 1/20 0.39
LRRK2 Q5S007 1/20 0.39
ALK Q9UM73 1/20 0.39
TYMP P19971 1/20 0.38
METAP2 P50579 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2870930 0.82 GAA (0.41) ALDH1A1CYP1A2CYP3A4NPC1SMN1; SMN2
SCHEMBL28021139 0.78 IDO1 (0.54) CYP2A6ALDH1A1CYP1A2CYP3A4BTK
SCHEMBL2876798 0.76 NT5E (0.42) SMN1; SMN2RXFP1IDO1FYN
SCHEMBL2875478 0.74 NOTUM (0.41) CYP1A2CYP3A4NPC1RAB9A
SCHEMBL16200078 0.73 MAPT (0.39) ALDH1A1CYP1A2CYP3A4SMN1; SMN2HSD17B10
SCHEMBL20837058 0.73 CYP2A6 (0.41) CYP2A6ALDH1A1CYP1A2CYP3A4BTK
SCHEMBL15660759 0.72 IDO1 (0.55) CYP2A6ALDH1A1CYP1A2CYP3A4BTK
SCHEMBL3464293 0.71 TDP1 (0.42) ALDH1A1CYP1A2BTKNPC1SMN1; SMN2
SCHEMBL2871119 0.69 NOTUM (0.37) RXFP1PIM1IDO1HSD17B10
SCHEMBL13683096 0.68 LMNA (0.46) CYP2A6ALDH1A1CYP1A2CYP3A4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed