SCHEMBL16200082

SCHEMBL16200082

COc1cccc(-c2[nH]nc(C)c2Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.47
ADORA1 P30542 5/20 0.47
NOTUM Q6P988 1/20 0.47
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
DCUN1D1 Q96GG9 1/20 0.47
DYRK1A Q13627 2/20 0.45
DYRK1B Q9Y463 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44
XDH P47989 1/20 0.43
HTR1A P08908 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR7 P34969 1/20 0.43
HTR2B P41595 1/20 0.43
HTR3A P46098 1/20 0.43
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5454847 0.77 CDC7 (0.49) NOTUMNR1H2NR1H3DCUN1D1DYRK1A
SCHEMBL2876858 0.77 AKT2 (0.50) GAASMN1; SMN2MAPTLMNAKDM4E
SCHEMBL13024563 0.76 GAA (0.55) ADORA2AADORA1NOTUMNR1H2NR1H3
SCHEMBL24765276 0.75 CHEK1 (0.59) NOTUMNR1H2NR1H3DCUN1D1DYRK1A
SCHEMBL8036864 0.74 NR1H2 (0.51) ADORA2AADORA1NOTUMNR1H2NR1H3
SCHEMBL8623261 0.71 MAPT (0.46) ADORA2ANOTUMNR1H2NR1H3DCUN1D1
SCHEMBL13426462 0.70 MAPT (0.61) NOTUMNR1H2NR1H3DCUN1D1DYRK1A
SCHEMBL17413462 0.70 NOTUM (0.54) NOTUMNR1H2NR1H3DCUN1D1DYRK1A
SCHEMBL29489425 0.70 CYP3A4 (0.73) NOTUMDYRK1ACLK4GAAXDH
SCHEMBL196765 0.70 CYP3A4 (0.73) NOTUMDYRK1ACLK4GAAXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed