SCHEMBL16200087

SCHEMBL16200087

CCc1ccc(Cl)c(SC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
SIGMAR1 Q99720 8/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2A6 P11509 1/20 0.38
MAPT P10636 4/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
IDO1 P14902 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17015131 0.77 KCNN4 (0.41) TRPA1SIGMAR1CYP1A2CYP2A6MAPT
SCHEMBL19574252 0.77 TRPA1 (0.40) TRPA1SIGMAR1CYP1A2CYP2A6MAPT
SCHEMBL11896057 0.75 SLC6A2 (0.40) TRPA1SIGMAR1CYP1A2CYP2A6MAPT
SCHEMBL93983 0.75 IDO1 (0.58) TRPA1SIGMAR1CYP1A2MAPTCYP2C19
SCHEMBL1145559 0.73 TP53 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19NPC1
SCHEMBL18922609 0.73 KMT2A (0.43) CYP1A2CYP2A6MAPTCYP3A4CYP2C9
Ammonia Solution, Strong SCHEMBL793693 0.73 IDO1 (0.56) TRPA1SIGMAR1CYP1A2MAPTCYP2C19
SCHEMBL12303991 0.72 TRPA1 (0.40) TRPA1CYP1A2CYP2A6MAPTCYP3A4
SCHEMBL3790563 0.71 TRPA1 (0.43) TRPA1SIGMAR1CYP1A2CYP2A6MAPT
SCHEMBL3789458 0.71 KMT2A (0.41) CYP1A2MAPTSMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed