SCHEMBL16211754

SCHEMBL16211754

O=C(O)N1CC(c2cc(Cl)nc(Cl)c2)C1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.36
S1PR2 O95136 1/20 0.36
SCD5 Q86SK9 7/20 0.35
SCD O00767 6/20 0.35
PROKR1 Q8TCW9 3/20 0.35
LMNA P02545 2/20 0.33
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
SPR P35270 2/20 0.33
NPC1 O15118 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16212231 0.84 FFAR1 (0.35) FFAR1S1PR2LMNA
SCHEMBL23089202 0.80 PROKR1 (0.49) SCD5SCDPROKR1
SCHEMBL15535023 0.77 MEN1 (0.42) TP53MAPT
SCHEMBL25255898 0.76 SCD5 (0.38) SCD5SCDPROKR1LMNATP53
SCHEMBL16211755 0.75 MAP3K12 (0.39) PROKR1LMNASPR
SCHEMBL162009 0.75 NAPRT (0.43) SMN1; SMN2TDP1
SCHEMBL23453444 0.74 SMN1; SMN2 (0.49) PROKR1LMNATP53MAPTNPC1
SCHEMBL16212243 0.73 MAP3K12 (0.37) PROKR1HSD11B1
SCHEMBL15535084 0.73 PROKR1 (0.43) PROKR1LMNASPRSMN1; SMN2HSD11B1
SCHEMBL18585817 0.72 HSD11B1 (0.53) LMNATP53MAPTSPRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991978-A1 BIHETEROARYL COMPOUNDS AND USES THEREOF F. Hoffmann-La Roche SA (CH) 2016-03-09 EP disclosed
WO-2014177060-A1 BIHETEROARYL COMPOUNDS AND USES THEREOF F.HOFFMANN-LA ROCHE AG (CH) 2014-11-06 WO disclosed