SCHEMBL16211981

SCHEMBL16211981

CC(C)(F)c1ccc(Cl)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.58
CYP3A4 P08684 2/20 0.58
TDP1 Q9NUW8 2/20 0.58
MAPK1 P28482 1/20 0.58
TP53 P04637 2/20 0.44
PDK2 Q15119 3/20 0.41
PDK1 Q15118 2/20 0.41
PDK3 Q15120 2/20 0.41
PDK4 Q16654 2/20 0.41
CASR P41180 1/20 0.40
HSD17B10 Q99714 2/20 0.39
PDE2A O00408 1/20 0.39
HSD11B1 P28845 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
CYP19A1 P11511 1/20 0.36
IDO1 P14902 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31740316 1.00 TSHR (0.58) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL107751 0.81 TSHR (0.62) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL29403188 0.81 TSHR (0.62) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL799844 0.81 TSHR (0.62) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL2270300 0.79 CYP3A4 (0.50) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL18243045 0.79 TSHR (0.60) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL21995301 0.79 TSHR (0.60) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL3654239 0.79 TSHR (0.60) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL3919506 0.78 CYP3A4 (0.48) TSHRCYP3A4TDP1MAPK1TP53
SCHEMBL16579369 0.77 TSHR (0.58) TSHRCYP3A4TDP1MAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3073827-A1 NEW PESTICIDAL COMPOUNDS AND USES Bayer Animal Health GmbH (DE) 2016-10-05 EP disclosed
EP-2991485-A1 N-(2-FLUORO-2-PHENETHYL)CARBOXAMIDES AS NEMATICIDES AND ENDOPARASITICIDES Bayer CropScience Aktiengesellschaft (DE) 2016-03-09 EP disclosed
WO-2015078800-A1 NEW PESTICIDAL COMPOUNDS AND USES BAYER CROPSCIENCE AG (DE) 2015-06-04 WO disclosed
WO-2014177582-A1 N-(2-FLUORO-2-PHENETHYL)CARBOXAMIDES AS NEMATICIDES AND ENDOPARASITICIDES BAYER CROPSCIENCE AG (DE) 2014-11-06 WO disclosed