SCHEMBL16229458

SCHEMBL16229458

CCCCCC(=O)Nc1ccc(NC(=S)NC(=O)c2cc(Cl)c(OC)c(Cl)c2)cc1

nearest known ligand 0.80

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 15/20 0.80
SIRT1 Q96EB6 12/20 0.80
TAS1R3 Q7RTX0 1/20 0.51
TAS1R1 Q7RTX1 1/20 0.51
TAS1R2 Q8TE23 1/20 0.51
CYP2C9 P11712 1/20 0.51
ALOX12 P18054 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229470 0.91 SIRT2 (0.85) SIRT2SIRT1
SCHEMBL16229460 0.91 SIRT2 (0.82) SIRT2SIRT1
SCHEMBL16229475 0.88 SIRT2 (0.63) SIRT2SIRT1CYP2C9ALOX12
Hydrochloric Acid SCHEMBL1706966 0.88 SIRT2 (0.98) SIRT2SIRT1
SCHEMBL16229459 0.88 SIRT2 (0.63) SIRT2SIRT1
SCHEMBL16229454 0.86 SIRT2 (0.78) SIRT2SIRT1
SCHEMBL16229472 0.85 SIRT2 (0.63) SIRT2SIRT1
Hydrochloric Acid SCHEMBL1706649 0.83 SIRT2 (0.98) SIRT2SIRT1
SCHEMBL16229381 0.82 SIRT1 (0.67) SIRT2SIRT1
SCHEMBL16229457 0.81 ALDH1A1 (0.65) SIRT2SIRT1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440522-B1 AROYLTHIOUREA AND ARYLTHIOCARBONYLUREA DERIVATIVES UNIV DUNDEE (GB) 2014-11-12 EP disclosed