SCHEMBL16229745

SCHEMBL16229745

CN1C2C1C21Cc2ccc(OCCNS(=O)(=O)CC3CC3)cc2C1Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 17/20 0.60
KCNH2 Q12809 2/20 0.57
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16784626 0.91 SLC6A9 (0.50) SLC6A9KCNH2MAOB
SCHEMBL16784655 0.91 SLC6A9 (0.50) SLC6A9KCNH2
SCHEMBL16229781 0.89 SLC6A9 (0.49) SLC6A9KCNH2SLC6A4
SCHEMBL16229747 0.87 SLC6A9 (0.43) SLC6A9KCNH2
SCHEMBL16229750 0.86 SLC6A9 (0.46) SLC6A9KCNH2MAOB
SCHEMBL16784624 0.86 SLC6A9 (0.46) SLC6A9KCNH2
SCHEMBL16784628 0.85 SLC6A9 (0.44) SLC6A9KCNH2
SCHEMBL16229752 0.82 SLC6A9 (0.52) SLC6A9KCNH2
SCHEMBL16229774 0.82 SLC6A9 (0.65) SLC6A9KCNH2
SCHEMBL16229782 0.80 SLC6A9 (0.39) SLC6A9KCNH2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed
US-8883839-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy ABBOTT LABORATORIES (US) 2014-11-11 US disclosed