SCHEMBL16239255

SCHEMBL16239255

O=C(NN1CCc2ccccc2C1)c1ccc(Br)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.55
NOD2 Q9HC29 1/20 0.55
NOD1 Q9Y239 1/20 0.55
LIPE Q05469 6/20 0.53
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
ALDH1A1 P00352 4/20 0.52
GAA P10253 3/20 0.52
HPGD P15428 2/20 0.52
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
MAPT P10636 2/20 0.46
HTT P42858 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14890641 0.88 LIPE (0.62) LIPENPC1RAB9AALDH1A1KMT2A
SCHEMBL14907137 0.86 LIPE (0.55) NOD1LIPENPC1RAB9AALDH1A1
SCHEMBL14907228 0.86 LIPE (0.66) TNFNOD2NOD1LIPEALDH1A1
SCHEMBL16238884 0.83 LIPE (0.51) LIPEHDAC6MAPT
SCHEMBL16239253 0.82 NPC1 (0.55) TNFNOD2NOD1LIPENPC1
SCHEMBL14890633 0.82 LIPE (0.73) TNFNOD2NOD1LIPENPC1
SCHEMBL20854509 0.80 AKR1C3 (0.43) TNFNOD2NOD1ALDH1A1GAA
SCHEMBL16251376 0.80 LIPE (0.50) TNFNOD2NOD1LIPENPC1
SCHEMBL7550712 0.80 LIPE (0.80) LIPENPC1RAB9AGAAMAPT
Benzenesulfonamide SCHEMBL16238901 0.79 CA1 (0.56) LIPEALDH1A1GAAHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889713-B1 N-substituted tetrahydroisoquinoline benzamides/benzene sulfonamides as anti-cancer agents FLORIDA A&M UNIVERSITY (US) 2014-11-18 US disclosed
US-8889713-B1 N-substituted tetrahydroisoquinoline benzamides/benzene sulfonamides as anti-cancer agents FLORIDA A&M UNIVERSITY (US) 2014-11-18 US disclosed