SCHEMBL16239697

SCHEMBL16239697

CN(C(=O)O)[C@@H]1CN(C(=O)c2ccc(C#N)cc2)C[C@@]1(C)c1ccc(Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 14/20 0.72
ALDH1A1 P00352 1/20 0.44
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
KDM1A O60341 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
HCRTR2 O43614 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10277847 0.84 TACR3 (1.00) TACR3
SCHEMBL16239850 0.82 TACR3 (0.75) TACR3
SCHEMBL16239536 0.79 TACR3 (0.74) TACR3ALDH1A1
SCHEMBL16239696 0.78 TACR3 (0.53) TACR3ALDH1A1NR1H4HCRTR2
SCHEMBL16239826 0.77 TACR3 (0.76) TACR3
SCHEMBL16239590 0.76 TACR3 (0.72) TACR3ALDH1A1
SCHEMBL16239794 0.73 TACR3 (0.71) TACR3
SCHEMBL16239848 0.73 TACR3 (0.71) TACR3
SCHEMBL16239606 0.72 TACR3 (0.62) TACR3
SCHEMBL16239673 0.71 TACR3 (0.73) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661432-B1 PYRROLIDINE DERIVATIVES AS NK3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed