SCHEMBL162434

SCHEMBL162434

CC[C@H](C)[C@](C)(N)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 2/20 0.34
GGT1 P19440 1/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34
TSHR P16473 2/20 0.33
KIF11 P52732 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
CYP2D6 P10635 2/20 0.32
ARG1 P05089 2/20 0.32
ARG2 P78540 2/20 0.32
CA2 P00918 2/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
GRM2 Q14416 1/20 0.32
GRM3 Q14832 1/20 0.32
CA1 P00915 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29489674 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL574079 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL22636108 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL202556 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL20854287 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL18274694 0.83 GABRR1 (0.36) ALDH1A1CYP1A2GGT1TSHRNOS1
SCHEMBL5322047 0.83 GABRR1 (0.36) ALDH1A1CYP1A2GGT1TSHRNOS1
SCHEMBL20854183 0.82 CHRM1 (0.44) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL20854296 0.82 CHRM1 (0.44) ALDH1A1CYP1A2GGT1MEN1THRB
SCHEMBL18770575 0.81 CA1 (0.35) KIF11CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2085 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250049970-A1 DLL3 TARGETING PEPTIDES AND CONSTRUCTS THEREOF MARIANA ONCOLOGY INC (US) 2025-02-13 US claimed
US-20250034210-A1 DLL3 TARGETING PEPTIDES AND CONSTRUCTS THEREOF MARIANA ONCOLOGY INC (US) 2025-01-30 US claimed
US-20250011368-A1 DLL3 TARGETING PEPTIDES AND CONSTRUCTS THEREOF MARIANA ONCOLOGY INC (US) 2025-01-09 US claimed
US-20160318987-A1 PROTEASE RESISTANT PEPTIDES MEDIMMUNE LIMITED (GB) 2016-11-03 US claimed
EP-3080153-A2 PROTEASE RESISTANT PEPTIDES Medimmune Limited (GB) 2016-10-19 EP claimed
WO-2015086686-A2 PROTEASE RESISTANT PEPTIDES MEDIMMUNE LIMITED (GB) 2015-06-18 WO claimed
US-20090215895-A1 Therapeutic and carrier molecules PEPLIN BIOLIPIDS PTY LTD (AU) 2009-08-27 US claimed
EP-1718602-A4 THERAPEUTIC AND CARRIER MOLECULES PEPLIN BIOLIPIDS PTY LTD (AU) 2007-12-12 EP claimed
US-7256172-B1 Method of treatment and agents useful for same THE UNIVERSITY OF MELBOURNE (AU) 2007-08-14 US claimed
EP-1718602-A1 THERAPEUTIC AND CARRIER MOLECULES Peplin Biolipids Pty Ltd. (AU) 2006-11-08 EP claimed
US-7070969-B1 Plasmin inhibitors from the australian brown snake Pseudonaja textilis textilis THE UNIVERSITY OF QUEENSLAND (AU) 2006-07-04 US claimed
WO-2005073164-A1 THERAPEUTIC AND CARRIER MOLECULES PEPLIN BIOLIPIDS PTY LTD (AU) 2005-08-11 WO claimed
WO-2026107423-A1 ORAL PEPTIDES AND USES THEREOF FOR WEIGHT LOSS, WEIGHT MAINTENANCE, AND MANAGEMENT OF METABOLIC CONDITIONS METSERA, INC. (US) 2026-05-21 WO disclosed
WO-2026085582-A1 PROTEIN CAGES THE UNIVERSITY OF SYDNEY (AU) 2026-04-30 WO disclosed
EP-4727655-A1 DLL3 TARGETING PEPTIDES AND CONSTRUCTS THEREOF Mariana Oncology Inc. (US) 2026-04-22 EP disclosed
US-20260069728-A1 MULTI-TARGETING COMPOUND AND USE THEREOF CHENGDU SHETAI MEDICAL TECHNOLOGY CO., LTD. (CN) 2026-03-12 US disclosed
WO-1994003483-A1 ENDOTHELIN RECEPTOR-BINDING COMPOUNDS CHIRON CORPORATION (US) 1994-02-17 WO disclosed
EP-0169300-B1 PROCESS FOR PREPARATION OF ALPHA-ALKYL AMINO ACIDS MERCK & CO. INC. (US) 1988-05-25 EP disclosed
EP-0169300-A1 Process for preparation of alpha-alkyl amino acids MERCK & CO. INC. (US) 1986-01-29 EP disclosed
US-4508921-A Process for preparation of alpha-alkyl amino acids MERCK & CO., INC. (US) 1985-04-02 US disclosed