SCHEMBL162470

SCHEMBL162470

COC(=O)CC(C)(C)Cc1ncc(-c2ccc(N)cc2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
CYP3A4 P08684 3/20 0.37
CSNK2A1 P68400 2/20 0.37
LOXL2 Q9Y4K0 2/20 0.37
PI4KB Q9UBF8 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 2/20 0.36
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
PDPK1 O15530 1/20 0.35
APP P05067 1/20 0.35
CSNK2A2 P19784 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL162291 0.85 XDH (0.43) ERCC5FEN1CSNK2A1ALDH1A1MAPT
SCHEMBL164309 0.82 ERCC5 (0.40) ERCC5FEN1CYP3A4CSNK2A1LOXL2
SCHEMBL160755 0.81 ERCC5 (0.41) ERCC5FEN1CYP3A4CSNK2A1LOXL2
SCHEMBL161347 0.81 DGAT1 (0.54) MAPTSMN1; SMN2LMNAHDAC6
SCHEMBL163569 0.80 PTPN1 (0.48) CSNK2A1SMN1; SMN2CSNK2A2
SCHEMBL161029 0.79 ERCC5 (0.39) ERCC5FEN1CYP3A4CSNK2A1LOXL2
SCHEMBL160763 0.78 DGAT1 (0.53) CYP3A4MAPTNPC1RAB9AMEN1
SCHEMBL164942 0.77 DGAT1 (0.55) MAPTNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL160848 0.77 ERCC5 (0.38) ERCC5FEN1CYP3A4CSNK2A1LOXL2
SCHEMBL163068 0.76 TRPV1 (0.45) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed