SCHEMBL6925668

SCHEMBL6925668

c1ccc(-c2c[nH]c(-c3ccc(N4CCCC4)nc3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.53
TSHR P16473 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
HPGD P15428 1/20 0.46
RECQL P46063 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 1/20 0.45
CNR1 P21554 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
FYN P06241 1/20 0.40
ATR Q13535 1/20 0.40
ADK P55263 1/20 0.40
AR P10275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6925885 0.99 CNR2 (0.56) CNR2TSHRNPC1RAB9AHPGD
SCHEMBL6924500 0.90 ATR (0.51) CNR2USP2HTTHSD17B10KDM4E
SCHEMBL6926900 0.88 CNR2 (0.53) CNR2TSHRHTTHSD17B10ALDH1A1
SCHEMBL6925451 0.88 FYN (0.54) FYNATR
SCHEMBL6927559 0.88 RAD52 (0.44) CNR2
SCHEMBL6926636 0.87 TSHR (0.46) CNR2TSHRNPC1RAB9AHPGD
SCHEMBL6928201 0.87 ADK (0.46) CNR2KMT2ALMNAKDM4EALDH1A1
SCHEMBL6925199 0.86 HRH3 (0.47) CNR2TSHRHPGDSMN1; SMN2USP2
SCHEMBL6920359 0.86 HRH3 (0.44) CNR2HPGDHSD17B10FYN
SCHEMBL6925622 0.85 HRH3 (0.45) HPGDSMN1; SMN2KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R CNR2 122/4885TSHR 227/4885NPC1 1762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.