SCHEMBL16260461

SCHEMBL16260461

COC(=O)c1cccc2c1Nc1ccccc1C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.58
TRPA1 O75762 4/20 0.49
LMNA P02545 2/20 0.44
TSHR P16473 2/20 0.44
ALDH1A1 P00352 2/20 0.42
CFTR P13569 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
ATM Q13315 1/20 0.41
AHR P35869 1/20 0.41
PDK2 Q15119 1/20 0.41
ROCK2 O75116 1/20 0.40
CSF1R P07333 1/20 0.40
KDR P35968 1/20 0.40
FLT3 P36888 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CDK5 Q00535 1/20 0.40
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23143494 0.88 ALOX5 (0.58) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL2445972 0.84 ALOX5 (0.45) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL2442681 0.84 ALOX5 (0.45) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL28085954 0.83 AHR (0.47) ALOX5ALDH1A1HSD17B10KDM4EAHR
SCHEMBL2447960 0.82 ALOX5 (0.43) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL2445893 0.82 ALOX5 (0.49) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL1639672 0.82 SMYD3 (0.53) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL14444038 0.81 ALOX5 (0.54) ALOX5TRPA1ALDH1A1HSD17B10KDM4E
SCHEMBL2442631 0.81 TRPA1 (0.45) ALOX5TRPA1LMNATSHRALDH1A1
SCHEMBL13425531 0.81 ALOX5 (0.47) ALOX5TRPA1LMNATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9356243-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2016-05-31 US disclosed
US-20140350243-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCH PATENT GMBH (DE) 2014-11-27 US disclosed