SCHEMBL16266166

SCHEMBL16266166

CC(C)(C)[Si](C)(C)OCc1sccc1-c1ccc2nc(-c3cnc4ccccc4c3)cn2c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A3 P47895 13/20 0.33
ALDH1A1 P00352 6/20 0.33
SLC2A1 P11166 1/20 0.33
ALDH1A2 O94788 1/20 0.33
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
ADORA2A P29274 1/20 0.32
NR4A2 P43354 1/20 0.32
KCNH2 Q12809 1/20 0.32
NPC1 O15118 3/20 0.31
PKM P14618 3/20 0.31
RAB9A P51151 3/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
MAPK1 P28482 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
KDM4E B2RXH2 2/20 0.30
TP53 P04637 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217714 0.84 ALDH1A3 (0.37) ALDH1A3ALDH1A1SLC2A1ALDH1A2PDGFRB
SCHEMBL3435794 0.70 NR4A2 (0.52) ALDH1A3ALDH1A1SLC2A1ALDH1A2PDGFRB
SCHEMBL217708 0.70 ALDH1A3 (0.42) ALDH1A3ALDH1A1SLC2A1ALDH1A2PDGFRB
Hydrochloric Acid SCHEMBL218759 0.69 ALDH1A3 (0.41) ALDH1A3ALDH1A1SLC2A1ALDH1A2PDGFRB
SCHEMBL3411468 0.68 NR4A2 (0.67) ALDH1A3ALDH1A1SLC2A1ALDH1A2NR4A2
SCHEMBL3430103 0.67 NR4A2 (0.39) ALDH1A3ALDH1A1SLC2A1ALDH1A2ADORA2A
SCHEMBL217710 0.66 NR4A2 (0.40) ALDH1A3ALDH1A1SLC2A1ALDH1A2PDGFRB
SCHEMBL3432955 0.66 NR4A2 (0.65) ALDH1A3ALDH1A1SLC2A1ALDH1A2NR4A2
SCHEMBL219947 0.66 L3MBTL1 (0.39) ALDH1A3ALDH1A1SLC2A1ALDH1A2NR4A2
SCHEMBL3430232 0.66 LRRK2 (0.39) ALDH1A1NR4A2NPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262804-B1 POLYSUBSTITUTED DERIVATIVES OF 6-HETEROARYL-IMIDAZO[L,2- A] PYRIDINES, AND PREPARATION AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2014-12-03 EP disclosed