SCHEMBL16299529

SCHEMBL16299529

CCCCC(=O)N1CCc2c([nH]c3ccc(Cl)cc23)C1c1ccc(C(=O)N2CCC(NC(C)=O)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 10/20 0.51
MAPT P10636 3/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 2/20 0.47
ABCG2 Q9UNQ0 4/20 0.46
ABCB1 P08183 1/20 0.44
TP53 P04637 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16299595 0.92 KIF11 (0.47) KIF11MAPTKDM4ELMNAABCG2
SCHEMBL765030 0.88 KIF11 (0.50) KIF11MAPTKDM4ELMNAABCG2
SCHEMBL8404507 0.75 KIF11 (0.47) KIF11MAPTLMNAABCG2ABCB1
SCHEMBL16359562 0.75 KIF11 (0.54) KIF11MAPTLMNATP53SMN1; SMN2
SCHEMBL8403171 0.75 KIF11 (0.49) KIF11MAPTKDM4ELMNAABCG2
SCHEMBL8403113 0.74 ALDH1A1 (0.50) KIF11MAPTKDM4ELMNAABCG2
SCHEMBL16313346 0.74 KIF11 (0.64) KIF11LMNAABCG2TP53SMN1; SMN2
SCHEMBL8403173 0.74 KIF11 (0.49) KIF11MAPTKDM4ELMNAABCG2
SCHEMBL3567366 0.74 KIF11 (0.74) KIF11MAPTLMNAABCG2
SCHEMBL16299551 0.74 KIF11 (0.53) KIF11MAPTLMNAABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871375-B1 CARBOLINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER PTC THERAPEUTICS INC (US) 2012-02-29 EP disclosed