SCHEMBL16299986

SCHEMBL16299986

CNC(=O)c1nc(OC)c(OC)c2c1CCN(Cc1ccc(F)c(Cl)c1)C2=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.40
POLB P06746 1/20 0.38
P2RX7 Q99572 13/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
TNIK Q9UKE5 1/20 0.35
AXL P30530 1/20 0.35
MERTK Q12866 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10232272 0.91 MEN1 (0.40) P2RX7ALDH1A1TNIKMEN1KMT2A
SCHEMBL10233464 0.91 MEN1 (0.36) P2RX7ALDH1A1TNIKMEN1KMT2A
SCHEMBL10232607 0.91 AKR1B1 (0.37) P2RX7TNIK
SCHEMBL2732419 0.88 PDPK1 (0.39) EGLN1P2RX7MEN1KMT2A
SCHEMBL10233800 0.84 PDPK1 (0.37) EGLN1POLBP2RX7MEN1KMT2A
SCHEMBL2734482 0.83 P2RX7 (0.34) P2RX7
SCHEMBL1335829 0.81 MEN1 (0.37) P2RX7ALDH1A1HTTMEN1KMT2A
SCHEMBL4481402 0.80 MEN1 (0.48) POLBALDH1A1HTTMEN1KMT2A
SCHEMBL4502946 0.79 AKR1B1 (0.43) EGLN1POLBALDH1A1HTTMEN1
SCHEMBL1336725 0.77 MEN1 (0.41) P2RX7ALDH1A1TNIKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058173-A1 HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed