SCHEMBL2734482

SCHEMBL2734482

COc1nc(C(=O)N2CCCC=C2C)c2c(c1OC)C(=O)N(Cc1ccc(F)c(Cl)c1)CC2

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 18/20 0.34
WDR5 P61964 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10232607 0.85 AKR1B1 (0.37) P2RX7
SCHEMBL10233464 0.85 MEN1 (0.36) P2RX7
SCHEMBL10232272 0.84 MEN1 (0.40) P2RX7
SCHEMBL16299986 0.83 EGLN1 (0.40) P2RX7
SCHEMBL1335829 0.78 MEN1 (0.37) P2RX7
SCHEMBL2732419 0.78 PDPK1 (0.39) P2RX7
SCHEMBL10233800 0.75 PDPK1 (0.37) P2RX7
SCHEMBL4502946 0.74 AKR1B1 (0.43) WDR5
SCHEMBL4481402 0.74 MEN1 (0.48)
SCHEMBL4483474 0.73 LMNA (0.45) WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632454-A1 HIV INTEGRASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058173-A1 HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed