SCHEMBL16301209

SCHEMBL16301209

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)NC(=O)OC(C)(C)C)C2)nc2cccc(OC)c21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.36
CYP2D6 P10635 4/20 0.36
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
KCNH2 Q12809 4/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
PADI4 Q9UM07 2/20 0.34
KLK5 Q9Y337 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GHSR Q92847 1/20 0.34
CHRM1 P11229 2/20 0.33
CASR P41180 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
TACR1 P25103 1/20 0.33
PPIA P62937 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763816 0.93 CTSB (0.36) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL763173 0.92 CTSB (0.35) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL741590 0.92 CTSB (0.35) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL741591 0.92 CTSB (0.35) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL762785 0.90 HRH1 (0.42) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL10293032 0.90 PADI4 (0.37) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL762600 0.89 HRH1 (0.40) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL763206 0.89 HRH1 (0.40) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL762559 0.88 KCNH2 (0.39) HRH1CYP2D6CTSBCTSSCTSK
SCHEMBL762548 0.87 KCNH2 (0.40) HRH1CYP2D6KCNH2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed