SCHEMBL16308170

SCHEMBL16308170

Cc1ccc2nc(C(F)F)n(-c3cc(N4CCOC[C@H]4C)nc(NCC4CCN(C5CCOCC5)CC4)n3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 7/20 0.42
CD274 Q9NZQ7 7/20 0.42
ATR Q13535 6/20 0.38
CHEK1 O14757 5/20 0.38
ATRIP Q8WXE1 5/20 0.38
PIK3CB P42338 3/20 0.37
PIK3CA P42336 7/20 0.36
PIK3R1 P27986 5/20 0.36
PIK3CD O00329 1/20 0.36
HTR4 Q13639 1/20 0.36
MTOR P42345 8/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15029298 0.91 PDCD1 (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL15029297 0.91 PDCD1 (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL15029348 0.90 PIK3CB (0.46) PIK3CBPIK3CAPIK3R1PIK3CDHTR4
SCHEMBL16308179 0.89 PDCD1 (0.43) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL15029787 0.89 PDCD1 (0.45) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL15029967 0.88 PDCD1 (0.43) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL16308152 0.85 PDCD1 (0.41) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL10125162 0.85 PDCD1 (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL10125164 0.85 PDCD1 (0.53) PDCD1CD274ATRCHEK1ATRIP
SCHEMBL16308183 0.84 PDCD1 (0.40) PDCD1CD274ATRCHEK1ATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2604601-B1 HETERO RING COMPOUND ASTELLAS PHARMA INC (JP) 2016-02-24 EP disclosed
US-8912180-B2 Heterocyclic compound ASTELLAS PHARMA INC. (JP) 2014-12-16 US disclosed
US-8912180-B2 Heterocyclic compound ASTELLAS PHARMA INC. (JP) 2014-12-16 US disclosed