SCHEMBL16312705

SCHEMBL16312705

Cc1ccn(Cc2ccc(OC(F)(F)F)cc2)c(=O)c1C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.47
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
MAPT P10636 4/20 0.44
TP53 P04637 2/20 0.44
CHRM5 P08912 3/20 0.43
MAPK14 Q16539 1/20 0.43
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
EPHX2 P34913 1/20 0.41
HCRTR1 O43613 3/20 0.41
HCRTR2 O43614 3/20 0.41
TYMS P04818 1/20 0.41
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE1C Q14123 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682507 0.86 GRM2 (0.46) GRM2LMNAALDH1A1TSHRMAPT
SCHEMBL1036013 0.77 GRM2 (0.54) GRM2LMNAALDH1A1TSHRMAPT
SCHEMBL1039732 0.77 GRM2 (0.54) GRM2LMNAALDH1A1TSHRMAPT
SCHEMBL171698 0.74 LMNA (0.51) GRM2LMNAALDH1A1MAPTHCRTR1
SCHEMBL18185700 0.74 PDE1C (0.51) GRM2LMNAALDH1A1TSHRMAPT
SCHEMBL2056309 0.74 ALDH1A1 (0.50) GRM2ALDH1A1TSHRCHRM5ABL1
SCHEMBL13047939 0.73 LMNA (0.51) GRM2LMNAMAPTTP53EPHX2
SCHEMBL169742 0.73 ALDH1A1 (0.44) GRM2LMNAALDH1A1TSHRCHRM5
SCHEMBL171738 0.73 ALDH1A1 (0.44) GRM2LMNAALDH1A1TSHRMAPT
SCHEMBL687245 0.72 GRM2 (0.43) GRM2LMNAALDH1A1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045836-B1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMA (US) 2008-03-05 EP disclosed