SCHEMBL16315186

SCHEMBL16315186

O=Nc1ccc(-n2ccc(-c3cccc(C(=O)O)c3)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPA1 P27694 1/20 0.43
STIM1 Q13586 6/20 0.42
ORAI1 Q96D31 6/20 0.42
KMO O15229 2/20 0.42
CD74 P04233 1/20 0.41
MIF P14174 1/20 0.41
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
MAP4K4 O95819 1/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
FGFR1 P11362 1/20 0.41
PRKACA P17612 1/20 0.41
KDR P35968 1/20 0.41
MAP2K2 P36507 1/20 0.41
MAPK8 P45983 1/20 0.41
CDK8 P49336 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL182162 0.86 KMO (0.53) RPA1STIM1ORAI1KMOCD74
SCHEMBL182038 0.85 RPA1 (0.45) RPA1STIM1ORAI1KMOCD74
SCHEMBL2708467 0.84 RPA1 (0.50) RPA1STIM1ORAI1KMOMAP4K4
SCHEMBL181876 0.84 KMT2A (0.51) RPA1STIM1ORAI1KMOCD74
SCHEMBL181928 0.84 HTT (0.52) RPA1STIM1ORAI1KMOCD74
SCHEMBL182136 0.84 KEAP1 (0.51) RPA1KMOCD74MIFNPC1
SCHEMBL182299 0.83 AURKA (0.53) RPA1STIM1ORAI1KMOCD74
SCHEMBL10194338 0.82 KDM5A (0.53) RPA1STIM1ORAI1KMOCD74
SCHEMBL181888 0.81 STIM1 (0.57) RPA1STIM1ORAI1NPC1RAB9A
SCHEMBL185371 0.81 KMT2A (0.49) STIM1ORAI1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2363129-A1 Pyrazole or triazole compounds and their use for the manufacture of a medicament for treating somatic mutation-related diseases PTC Therapeutics, Inc. (US) 2011-09-07 EP disclosed