SCHEMBL16319189

SCHEMBL16319189

CC(C)(C)[Si](C)(C)Oc1ccc(Br)c(CC2(C#N)CCCC2)c1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.37
CA1 P00915 4/20 0.37
CA9 Q16790 4/20 0.37
PREP P48147 3/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318652 0.79 SMN1; SMN2 (0.32) CA12CA1CA9BACE1
SCHEMBL16319169 0.77 BACE1 (0.33) BACE1
SCHEMBL16319029 0.75 CA12 (0.39) CA12CA1CA9PREP
SCHEMBL2292629 0.73 CA12 (0.44) CA12CA1CA9PREP
SCHEMBL14110450 0.73 CA12 (0.48) CA12CA1CA9PREP
SCHEMBL2188571 0.72 CA12 (0.43) CA12CA1CA9PREP
SCHEMBL9034920 0.72 CA12 (0.43) CA12CA1CA9PREP
SCHEMBL15690979 0.69 CA12 (0.43) CA12CA1CA9PREP
SCHEMBL17923729 0.69 PREP (0.41) CA12CA1CA9PREP
SCHEMBL25227167 0.68 ALDH1A1 (0.43) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed