SCHEMBL16319169

SCHEMBL16319169

COc1ccc(F)c(-c2ccc(O[Si](C)(C)C(C)(C)C)cc2CC2(C#N)CCC2)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
FFAR1 O14842 7/20 0.32
APP P05067 1/20 0.31
PROKR1 Q8TCW9 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318652 0.98 SMN1; SMN2 (0.32) BACE1SMN1; SMN2NPSR1FFAR1APP
SCHEMBL16319294 0.82 FFAR1 (0.36) FFAR1
SCHEMBL16319289 0.80 FFAR1 (0.34) SMN1; SMN2NPSR1FFAR1MEN1MAPT
SCHEMBL16319250 0.80 FFAR1 (0.36) FFAR1
SCHEMBL16318905 0.80 FFAR1 (0.33) NPSR1FFAR1MEN1MAPTKMT2A
SCHEMBL16318804 0.79 FFAR1 (0.35) FFAR1
SCHEMBL16318844 0.78 FFAR1 (0.42) FFAR1
SCHEMBL16319189 0.77 CA12 (0.37) BACE1
SCHEMBL16318884 0.76 FFAR1 (0.35) FFAR1
SCHEMBL16319117 0.71 CNR1 (0.35) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382188-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-05 US disclosed
EP-2816023-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed