SCHEMBL16319308

SCHEMBL16319308

CS(=O)(=O)NC(=O)c1c(F)cc(Oc2ccc(Cl)c(C(F)(F)F)c2)c(F)c1F

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.59
SCN5A Q14524 2/20 0.52
PLA2G7 Q13093 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370953 0.90 SCN9A (0.55) SCN9ASCN5A
SCHEMBL16319523 0.87 SCN9A (0.56) SCN9ASCN5A
SCHEMBL369786 0.84 SCN9A (0.81) SCN9ASCN5A
SCHEMBL16319537 0.84 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16319584 0.84 SCN9A (0.60) SCN9ASCN5APLA2G7
SCHEMBL680215 0.82 SCN9A (0.69) SCN9ASCN5A
SCHEMBL16319404 0.82 SCN9A (0.53) SCN9APLA2G7
SCHEMBL16319499 0.82 SCN9A (0.63) SCN9ASCN5APLA2G7
SCHEMBL16319431 0.82 SCN9A (0.68) SCN9ASCN5A
SCHEMBL680188 0.81 SCN9A (0.59) SCN9ASCN5APLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed