SCHEMBL16319499

SCHEMBL16319499

CS(=O)(=O)NC(=O)c1ccc(Oc2ccc(Cl)c(C(F)(F)F)c2)c(F)c1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 17/20 0.63
SCN5A Q14524 2/20 0.63
PLA2G7 Q13093 2/20 0.47
MRGPRX4 Q96LA9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319487 0.91 SCN9A (0.65) SCN9ASCN5APLA2G7MRGPRX4
SCHEMBL16319828 0.88 SCN9A (0.70) SCN9ASCN5A
SCHEMBL16319310 0.88 SCN9A (0.71) SCN9ASCN5A
SCHEMBL16319454 0.87 SCN9A (0.60) SCN9ASCN5APLA2G7
SCHEMBL371116 0.87 SCN9A (0.67) SCN9ASCN5A
SCHEMBL16319655 0.86 PLA2G7 (0.62) SCN9ASCN5APLA2G7
SCHEMBL16319431 0.85 SCN9A (0.68) SCN9ASCN5A
SCHEMBL16319537 0.85 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16319531 0.85 SCN9A (0.58) SCN9ASCN5AMRGPRX4
SCHEMBL16319394 0.83 SCN9A (0.66) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed