SCHEMBL16319578

SCHEMBL16319578

CS(=O)(=O)NC(=O)c1cc(F)c(Oc2ccc(C#N)c(Cl)c2)cc1F

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.77
SCN5A Q14524 2/20 0.53
SCN2B O60939 1/20 0.50
SCN1A P35498 1/20 0.50
SCN1B Q07699 1/20 0.50
PGR P06401 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16319598 0.87 SCN9A (1.00) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16319330 0.85 SCN9A (0.83) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16319641 0.85 SCN9A (0.87) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL679781 0.84 SCN9A (0.67) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16319304 0.83 SCN9A (0.58) SCN9ASCN5A
SCHEMBL16240228 0.83 SCN9A (0.78) SCN9ASCN5A
SCHEMBL16319485 0.83 SCN9A (0.83) SCN9ASCN5A
SCHEMBL679946 0.82 SCN9A (0.78) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16319777 0.82 SCN9A (0.78) SCN9ASCN5ASCN2BSCN1ASCN1B
SCHEMBL16319336 0.82 SCN9A (0.55) SCN9ASCN5ASCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed