SCHEMBL16334362

SCHEMBL16334362

COc1ccc(CSc2ncccc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.51
HPGD P15428 2/20 0.46
CLK4 Q9HAZ1 1/20 0.46
SYK P43405 2/20 0.46
AURKB Q96GD4 1/20 0.46
INCENP Q9NQS7 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
PKM P14618 1/20 0.45
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
SLC29A1 Q99808 1/20 0.43
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 1/20 0.43
APP P05067 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26964190 0.94 TP53 (0.49) TP53HPGDSYKAURKBINCENP
SCHEMBL16334229 0.85 TP53 (0.44) TP53HPGDSYKL3MBTL1PKM
SCHEMBL16334791 0.83 FFAR4 (0.49) TP53HPGDCLK4SYKAURKB
SCHEMBL26964234 0.82 TP53 (0.53) TP53HPGDL3MBTL1PKMALDH1A1
SCHEMBL16334065 0.81 TP53 (0.52) TP53HPGDL3MBTL1PKMALDH1A1
SCHEMBL2099509 0.81 TP53 (0.52) TP53HPGDL3MBTL1PKMALDH1A1
SCHEMBL16334749 0.80 SYK (0.46) TP53HPGDCLK4SYKAURKB
SCHEMBL10414873 0.79 ALDH1A1 (0.58) TP53L3MBTL1PKMALDH1A1SMN1; SMN2
SCHEMBL26964197 0.77 TP53 (0.48) TP53HPGDL3MBTL1PKMALDH1A1
SCHEMBL16334706 0.77 FFAR4 (0.53) HPGDCLK4SYKAURKBINCENP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105392777-B Biaryl derivatives as GPR120 agonists 株式会社LG化学 2020-09-22 CN disclosed
EP-3013796-B9 BIARYL DERIVATIVES AS GPR120 AGONISTS LG CHEMICAL LTD (KR) 2020-07-01 EP disclosed
EP-3628661-A1 BIARYL DERIVATIVES AS GPR120 AGONISTS LG CHEM, LTD. (KR) 2020-04-01 EP disclosed
US-10221138-B2 Biaryl derivatives as GPR120 agonists LG CHEM, LTD. (KR) 2019-03-05 US disclosed
US-20160168096-A1 BIARYL DERIVATIVES AS GPR120 AGONISTS LG LIFE SCIENCES LTD. (KR) 2016-06-16 US disclosed
EP-3013796-A1 BIARYL DERIVATIVES AS GPR120 AGONISTS LG Life Sciences Ltd. (KR) 2016-05-04 EP disclosed
WO-2014209034-A1 BIARYL DERIVATIVES AS GPR120 AGONISTS LG LIFE SCIENCES LTD. (KR) 2014-12-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160168096-A1 BIARYL DERIVATIVES AS GPR120 AGONISTS GPR119, GLP1R, GIPR TP53 4800/4885HPGD 2858/4885CLK4 3077/4885
US-10221138-B2 Biaryl derivatives as GPR120 agonists GPR119, GLP1R, GIPR TP53 4800/4885HPGD 2858/4885CLK4 3077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.