SCHEMBL16339677

SCHEMBL16339677

Ic1ccc(NN=Cc2ccccc2)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 1/20 0.50
NOX1 Q9Y5S8 1/20 0.49
RAB9A P51151 12/20 0.48
NPC1 O15118 9/20 0.48
MAPT P10636 6/20 0.48
GAA P10253 3/20 0.48
CASP3 P42574 2/20 0.48
SENP7 Q9BQF6 2/20 0.48
SENP6 Q9GZR1 2/20 0.48
MAPK1 P28482 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 6/20 0.47
KMT2A Q03164 6/20 0.47
SMN1; SMN2 Q16637 6/20 0.46
CDK5 Q00535 2/20 0.46
CDK5R1 Q15078 2/20 0.46
GFER P55789 1/20 0.46
LMNA P02545 2/20 0.46
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16339676 1.00 CYP1A2 (0.50) CYP1A2CYP3A4NOX1RAB9ANPC1
SCHEMBL12050032 0.81 RAB9A (0.63) CYP1A2CYP3A4NOX1RAB9ANPC1
SCHEMBL14638987 0.80 NPC1 (0.56) CYP1A2CYP3A4RAB9ANPC1MAPT
SCHEMBL16218785 0.80 NPC1 (0.56) CYP1A2CYP3A4RAB9ANPC1MAPT
SCHEMBL14638988 0.80 NPC1 (0.56) CYP1A2CYP3A4RAB9ANPC1MAPT
Hydrochloric Acid SCHEMBL11640901 0.79 CYP1A2 (0.49) CYP1A2CYP3A4NOX1RAB9ANPC1
Hydrochloric Acid SCHEMBL11640898 0.79 CYP1A2 (0.49) CYP1A2CYP3A4NOX1RAB9ANPC1
Hydrochloric Acid SCHEMBL11641096 0.78 CYP1A2 (0.48) CYP1A2CYP3A4NOX1RAB9ANPC1
Hydrochloric Acid SCHEMBL11641098 0.78 CYP1A2 (0.48) CYP1A2CYP3A4NOX1RAB9ANPC1
SCHEMBL1357771 0.77 RAB9A (0.72) CYP1A2CYP3A4RAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2818471-A1 Nitrogen bicyclic compounds as inhibitors for Scyl1 and Grk5 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-12-31 EP disclosed