SCHEMBL16349367

SCHEMBL16349367

COC(C)(C)c1cncn1C

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.34
CYP17A1 P05093 1/20 0.34
IDO1 P14902 1/20 0.31
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14253920 0.77 RORC (0.32) CYP3A4CYP17A1RORC
SCHEMBL14253919 0.72 RORC (0.33) CYP3A4CYP17A1RORC
SCHEMBL13813431 0.71 CYP3A4 (0.34) CYP3A4CYP17A1IDO1RORC
SCHEMBL14253917 0.71 CYP17A1 (0.34) CYP3A4CYP17A1IDO1RORC
SCHEMBL25289009 0.67 CYP17A1 (0.43) CYP3A4CYP17A1IDO1RORC
SCHEMBL13813446 0.64 TSHR (0.34)
SCHEMBL21573048 0.63 RORC (0.37) CYP3A4CYP17A1RORC
SCHEMBL21719301 0.63 TBXAS1 (0.35) CYP3A4CYP17A1RORC
SCHEMBL22388552 0.63 TBXAS1 (0.35) CYP3A4CYP17A1RORC
SCHEMBL24092913 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7342016-B2 Farnesyl protein transferase inhibitors as antitumor agents SCHERING CORPORATION (US) 2008-03-11 US disclosed