SCHEMBL16360425

SCHEMBL16360425

CC(=O)CNc1ccc(CC(N)C(C)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSK P41240 1/20 0.43
SLC7A5 Q01650 2/20 0.42
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
PTPRC P08575 1/20 0.38
CA12 O43570 5/20 0.37
CA1 P00915 5/20 0.37
CA2 P00918 5/20 0.37
CA7 P43166 5/20 0.37
TDP1 Q9NUW8 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
TPH1 P17752 1/20 0.36
GRB2 P62993 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12155049 0.89 SLC7A5 (0.57) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL826519 0.89 SLC7A5 (0.57) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL15081041 0.86 ALDH1A1 (0.46) CSKSLC7A5ALPIPKMPTGS1
SCHEMBL19733539 0.81 SLC7A5 (0.46) CSKSLC7A5ALPIPKMPTGS1
SCHEMBL7471913 0.77 ALDH1A1 (0.52) CA12CA1CA2CA7TDP1
SCHEMBL14355742 0.77 SLC7A5 (0.48) CSKSLC7A5ALPIPKMPTGS1
SCHEMBL14559931 0.77 SLC7A5 (0.48) CSKSLC7A5ALPIPKMPTGS1
SCHEMBL9780166 0.77 SLC7A5 (0.59) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL26747607 0.75 ITGB3 (0.41) CSKSLC7A5ALPIPKMPTGS1
SCHEMBL12028154 0.75 SLC7A5 (0.53) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012166560-A1 COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES AMBRX, INC. (US) 2012-12-06 WO disclosed