SCHEMBL16370488

SCHEMBL16370488

CCOC(=O)c1nc(-c2ccccc2)ns1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.59
L3MBTL1 Q9Y468 3/20 0.59
SMN1; SMN2 Q16637 8/20 0.52
RAB9A P51151 7/20 0.52
LMNA P02545 5/20 0.52
MAPT P10636 3/20 0.52
KDM4E B2RXH2 3/20 0.52
TP53 P04637 3/20 0.52
HSD17B10 Q99714 2/20 0.52
MAPK1 P28482 1/20 0.52
ATM Q13315 1/20 0.52
NPC1 O15118 6/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HTT P42858 1/20 0.51
CDC7 O00311 1/20 0.50
TRPM8 Q7Z2W7 1/20 0.50
DBF4 Q9UBU7 1/20 0.50
RARA P10276 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4114732 0.88 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTKDM4ETP53
SCHEMBL14527733 0.87 ALDH1A1 (0.45) ALDH1A1L3MBTL1RAB9ALMNAMAPT
SCHEMBL1425593 0.86 ALDH1A1 (0.51) ALDH1A1L3MBTL1LMNAMEN1KMT2A
SCHEMBL1426050 0.86 MAPT (0.52) ALDH1A1L3MBTL1SMN1; SMN2RAB9ALMNA
SCHEMBL18614346 0.86 MAPT (0.54) ALDH1A1L3MBTL1SMN1; SMN2RAB9ALMNA
SCHEMBL1425605 0.85 MAPT (0.61) ALDH1A1L3MBTL1SMN1; SMN2RAB9ALMNA
SCHEMBL21348642 0.84 TDP1 (0.53) ALDH1A1L3MBTL1SMN1; SMN2RAB9ALMNA
SCHEMBL4164682 0.84 FOS (0.46) ALDH1A1L3MBTL1RAB9ALMNAMAPT
SCHEMBL4101439 0.83 PPARD (0.44) ALDH1A1L3MBTL1SMN1; SMN2RAB9ALMNA
SCHEMBL4114734 0.82 MAPT (0.55) ALDH1A1L3MBTL1MAPTKDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12433895-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2025-10-07 US disclosed
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE PHARMARESROUCES (SHANGHAI) CO., LTD. (CN) 2024-10-10 US disclosed
US-11844758-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2023-12-19 US disclosed
CN-111087353-B Therapeutically active compounds and methods of use thereof 法国施维雅药厂 2023-10-24 CN disclosed
US-20220354856-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2022-11-10 US disclosed
US-10946023-B2 Therapeutically active compounds and their methods of use AGIOS PHARMACEUTICALS, INC. (US) 2021-03-16 US disclosed
US-10946023-B2 Therapeutically active compounds and their methods of use AGIOS PHARMACEUTICALS, INC. (US) 2021-03-16 US disclosed
EP-3686190-A1 SYNTHESIS OF THERAPEUTICALLY ACTIVE COMPOUNDS Agios Pharmaceuticals, Inc. (US) 2020-07-29 EP disclosed
CN-111087353-A Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2020-05-01 CN disclosed
CN-105473560-B Therapeutically active compounds and methods of use thereof 安吉奥斯医药品有限公司 2020-01-17 CN disclosed
US-20170107194-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2017-04-20 US disclosed
US-20170107194-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2017-04-20 US disclosed
US-9579324-B2 Therapeutically active compounds and their methods of use AGIOS PHARMACEUTICALS, INC (US) 2017-02-28 US disclosed
US-9579324-B2 Therapeutically active compounds and their methods of use AGIOS PHARMACEUTICALS, INC (US) 2017-02-28 US disclosed
US-9579324-B2 Therapeutically active compounds and their methods of use AGIOS PHARMACEUTICALS, INC (US) 2017-02-28 US disclosed
US-20160220572-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2016-08-04 US disclosed
US-20160220572-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2016-08-04 US disclosed
US-20160220572-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2016-08-04 US disclosed
EP-3019483-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE Agios Pharmaceuticals, Inc. (US) 2016-05-18 EP disclosed
WO-2015003640-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE AGIOS PHARMACEUTICALS, INC. (US) 2015-01-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12433895-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-11844758-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-10946023-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-20160220572-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-20170107194-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885
US-20220354856-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT ALDH1A1 923/4885L3MBTL1 1106/4885SMN1; SMN2 568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.